Nicotinic Acetylcholine Receptors

Peptide neurotoxins, small-cell lung carcinoma andneurological paraneoplastic syndromes

Neurology / Immune response / Ion Channels / Antibodies / Humans / Hormones / Nicotinic Acetylcholine Receptors / Non small cell carcinoma / Neurotoxins / Biochimie / Paraneoplastic Syndromes / Calcium Ions / Biochemistry and cell biology / Calcium Channel Blockers / Hormones / Nicotinic Acetylcholine Receptors / Non small cell carcinoma / Neurotoxins / Biochimie / Paraneoplastic Syndromes / Calcium Ions / Biochemistry and cell biology / Calcium Channel Blockers

The peroxisome proliferator activated receptor regulates malic enzyme gene expression

Immunology / Stem Cells / Kinetics / Mitochondria / Immunology of the Gut / Biological Chemistry / Transcription Factors / Molecular endocrinology / Gene expression / Multidisciplinary / Western blotting / Biological Sciences / DNA / RNA interference / Cell Differentiation / Molecular and cellular biology / Humans / Endothelial Cells / Fatty acids / Mice / G protein-coupled receptors / Animals / Male / Nicotinic Acetylcholine Receptors / RETINOIDS / Adipogenesis / Peroxisome proliferator-activated receptor / Lipid metabolism / Triglycerides / Clinical Sciences / CHEMICAL SCIENCES / Rats / Oxygen / Chromatin Immunoprecipitation / Oral Hypoglycemic Agents / Adipocytes / Peroxisome / Body Weight / Veterinary Sciences / Thiazoles / Base Sequence / Recombinant Proteins / Retinal Diseases / Protein Binding / #Hypolipidemic Agents / Gene Expression Regulation / Biological Chemistry / Transcription Factors / Molecular endocrinology / Gene expression / Multidisciplinary / Western blotting / Biological Sciences / DNA / RNA interference / Cell Differentiation / Molecular and cellular biology / Humans / Endothelial Cells / Fatty acids / Mice / G protein-coupled receptors / Animals / Male / Nicotinic Acetylcholine Receptors / RETINOIDS / Adipogenesis / Peroxisome proliferator-activated receptor / Lipid metabolism / Triglycerides / Clinical Sciences / CHEMICAL SCIENCES / Rats / Oxygen / Chromatin Immunoprecipitation / Oral Hypoglycemic Agents / Adipocytes / Peroxisome / Body Weight / Veterinary Sciences / Thiazoles / Base Sequence / Recombinant Proteins / Retinal Diseases / Protein Binding / #Hypolipidemic Agents / Gene Expression Regulation

3-(5-Alkylamino-4-isoxazolyl)-1,2,5,6-tetrahydropyridines: a novel class of central nicotinic receptor ligands

Organic Chemistry / Mass Spectrometry / Magnetic Resonance Spectroscopy / Cerebral Cortex / Animals / Male / Nicotinic Acetylcholine Receptors / Rats / Pyridines / Wistar Rats / Bioorganic and medicinal Chemistry / Muscarinic Receptor / Ligands / Male / Nicotinic Acetylcholine Receptors / Rats / Pyridines / Wistar Rats / Bioorganic and medicinal Chemistry / Muscarinic Receptor / Ligands

A  induces astrocytic glutamate release, extrasynaptic NMDA receptor activation, and synaptic loss

Multidisciplinary / Fluorescence Resonance Energy Transfer / Transgenic Mice / Hippocampus / Glutamate / Humans / Mice / Female / Animals / Male / Nicotinic Acetylcholine Receptors / Astrocyte / Acetylcholine / Whole cell recording / Astrocytes / Synaptic Depression / Rats / SYNAPSES / Cognitive Decline / Alzheimer Disease / Glutamic Acid / Humans / Mice / Female / Animals / Male / Nicotinic Acetylcholine Receptors / Astrocyte / Acetylcholine / Whole cell recording / Astrocytes / Synaptic Depression / Rats / SYNAPSES / Cognitive Decline / Alzheimer Disease / Glutamic Acid

Synthesis and pharmacological characterization of 5-phenyl-2-[2-(1-piperidinylcarbonyl)phenyl]-2,3-dihydro-1 H-pyrrolo[1,2- c]imidazol-1-ones: A new class of Neuropeptide S antagonists

Inorganic Chemistry / Organic Chemistry / Medicinal Chemistry / Calcium / Pharmaceutical Chemistry / Macromolecular X-Ray Crystallography / Patch-clamp and imaging techniques / Dogs / Cell line / Adenosine / Brain / Humans / Discrimination Learning / Cerebral Cortex / Mice / Nicotine / Animals / Male / Nicotinic Acetylcholine Receptors / Organometallics / Neurons / CHEMICAL SCIENCES / Rats / Radioligand Assay / Pyridines / BIOCHEMICAL PHARMACOLOGY / Molecular Conformation / Protein Conformation / Alanine / Bioorganic and medicinal Chemistry / Radiopharmaceuticals / Rabbits / Structure activity Relationship / Recombinant Proteins / Ligands / Pain Measurement / Monte Carlo Method / Analgesics / Molecular Structure / Macromolecular X-Ray Crystallography / Patch-clamp and imaging techniques / Dogs / Cell line / Adenosine / Brain / Humans / Discrimination Learning / Cerebral Cortex / Mice / Nicotine / Animals / Male / Nicotinic Acetylcholine Receptors / Organometallics / Neurons / CHEMICAL SCIENCES / Rats / Radioligand Assay / Pyridines / BIOCHEMICAL PHARMACOLOGY / Molecular Conformation / Protein Conformation / Alanine / Bioorganic and medicinal Chemistry / Radiopharmaceuticals / Rabbits / Structure activity Relationship / Recombinant Proteins / Ligands / Pain Measurement / Monte Carlo Method / Analgesics / Molecular Structure

A  induces astrocytic glutamate release, extrasynaptic NMDA receptor activation, and synaptic loss

Multidisciplinary / Fluorescence Resonance Energy Transfer / Transgenic Mice / Hippocampus / Glutamate / Humans / Mice / Female / Animals / Male / Nicotinic Acetylcholine Receptors / Astrocyte / Acetylcholine / Whole cell recording / Astrocytes / Synaptic Depression / Rats / SYNAPSES / Cognitive Decline / Alzheimer Disease / Glutamic Acid / Humans / Mice / Female / Animals / Male / Nicotinic Acetylcholine Receptors / Astrocyte / Acetylcholine / Whole cell recording / Astrocytes / Synaptic Depression / Rats / SYNAPSES / Cognitive Decline / Alzheimer Disease / Glutamic Acid

Temporal coherency between receptor expression, neural activity and AP-1-dependent transcription regulates Drosophila motoneuron dendrite development

Fluorescence Microscopy / Immunohistochemistry / Drosophila melanogaster / Confocal Microscopy / Development / Signal Transduction / Biological Sciences / Animals / Nicotinic Acetylcholine Receptors / Dendrites / Synaptic Transmission / Cell nucleus / Time Factors / Signal Transduction / Biological Sciences / Animals / Nicotinic Acetylcholine Receptors / Dendrites / Synaptic Transmission / Cell nucleus / Time Factors

5α-Cardenolides from Kanahia laniflora Inhibit Ionotropic Acetylcholine Receptors

Complementary and Alternative Medicine / Plant Biology / Pharmacognosy / Patch-clamp and imaging techniques / Phytotherapy / Humans / Nicotinic Acetylcholine Receptors / Flowers / Plant extracts / Cholinergic Receptor / Apocynaceae / Plant Leaves / Humans / Nicotinic Acetylcholine Receptors / Flowers / Plant extracts / Cholinergic Receptor / Apocynaceae / Plant Leaves

Traumatic Brain Injury Elicits Similar Alterations in α7 Nicotinic Receptor Density in Two Different Experimental Models

Traumatic Brain Injury / Drug development / Brain / Humans / Child / Female / Animals / Male / Nicotinic Acetylcholine Receptors / Young Adult / Clinical Sciences / Rats / Swine / Autoradiography / Survival Time / Neurosciences / Experimental Model / Brain injuries / Random Allocation / Female / Animals / Male / Nicotinic Acetylcholine Receptors / Young Adult / Clinical Sciences / Rats / Swine / Autoradiography / Survival Time / Neurosciences / Experimental Model / Brain injuries / Random Allocation
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